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Instruction of (2R)-2-(4-Hydroxyphenyl)glycyl-N-[(2S,5R,6R)-2-carboxy-3,3-dimethyl-7-oxo-4-thia-1-azabicyclo[3.
2.
0]hept-6-yl]-(2R)-2-(4-hydroxyphenyl)glycinamide: A Comprehensive Guide
In the field of pharmaceuticals, the discovery and development of new drugs is a constant and ongoing process.
This requires a thorough understanding of the underlying mechanisms of disease and the use of innovative chemical synthesis techniques to create new compounds with potential therapeutic benefits.
One such compound is (2R)-2-(4-Hydroxyphenyl)glycyl-N-[(2S,5R,6R)-2-carboxy-3,3-dimethyl-7-oxo-4-thia-1-azabicyclo[3.
2.
0]hept-6-yl]-(2R)-2-(4-hydroxyphenyl)glycinamide, which has shown promise in pre-clinical trials for the treatment of several diseases.
This article aims to provide a comprehensive guide to the synthesis and production of (2R)-2-(4-Hydroxyphenyl)glycyl-N-[(2S,5R,6R)-2-carboxy-3,3-dimethyl-7-oxo-4-thia-1-azabicyclo[3.
2.
0]hept-6-yl]-(2R)-2-(4-hydroxyphenyl)glycinamide.
This will include an overview of the chemical reaction mechanisms involved in the synthesis of the compound, as well as the key steps in the production process.
Synthesis of (2R)-2-(4-Hydroxyphenyl)glycyl-N-[(2S,5R,6R)-2-carboxy-3,3-dimethyl-7-oxo-4-thia-1-azabicyclo[3.
2.
0]hept-6-yl]-(2R)-2-(4-hydroxyphenyl)glycinamide
The synthesis of (2R)-2-(4-Hydroxyphenyl)glycyl-N-[(2S,5R,6R)-2-carboxy-3,3-dimethyl-7-oxo-4-thia-1-azabicyclo[3.
2.
0]hept-6-yl]-(2R)-2-(4-hydroxyphenyl)glycinamide involves a multi-step synthesis process.
The following is a general overview of the key steps involved in the synthesis of this compound:
Step 1: Synthesis of 4-[(2,4-dimethoxyphenyl)methylene]-2-oxo-1,3-oxazolidin-3-one
The synthesis of 4-[(2,4-dimethoxyphenyl)methylene]-2-oxo-1,3-oxazolidin-3-one involves the reaction of 2,4-dimethoxybenzaldehyde with methyl 4-oxo-4H-1,3-oxazidine-3-carboxylate to form the desired product.
Step 2: Synthesis of 2-[(2,4-dimethoxyphenyl)methyleneamino]-N-(4-methoxy-3-oxo-2H-1,2,3-benzoxadiazid-7-yl)-acetamide
The synthesis of 2-[(2,4-dimethoxyphenyl)methyleneamino]-N-(4-methoxy-3-oxo-2H-1,2,3-benzoxadiazid-7-yl)-acetamide involves the reaction of 4-methoxy-3-oxo-2H-1,2,3-benzoxadiazide-7-ylamine with 2-chloro-N-(2,4-dimethoxyphenyl)acetamide to form the desired product.
Step 3: Synthesis of N